Co-Target(s) Information

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Target General Information
Co-Targets of This Target
References
Target General Information  Top
Target ID T32262 Target Info
Target Name Calcitonin gene-related peptide receptor (CGRPR)
Synonyms
Calcitonin receptor-like receptor; Calcitonin gene-related peptide type 1 receptor; CGRPR; CGRP type 1 receptor
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Target Type Successful Target
Gene Name CALCRL
Biochemical Class GPCR secretin
UniProt ID
CALRL_HUMAN
Co-Targets of This Target  Top
Co-Target Name Calcitonin gene-related peptide 1 (CALCA) Clinical trial Target
UniProt ID CALCA_HUMAN
Gene Name CALCA
Synonyms
Calcitonin gene-related peptide I; CGRP-I; CALCA; CALC1; Alpha-type CGRP
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Representative Drug(s) Olcegepant Drug Info Ki = 0.014 nM Click to Show More [1]
2 MK-3207 Drug Info Ki = 0.024 nM [1]
3 Telcagepant Drug Info Ki = 0.78 nM [1]
References  Top
REF 1 Identification of a novel RAMP-independent CGRP receptor antagonist. Bioorg Med Chem Lett. 2011 Nov 15;21(22):6705-8.

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