Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T16633 | Target Info | |||
| Target Name | Somatostatin receptor type 1 (SSTR1) | ||||
| Synonyms |
Sst(1); Somatostatin receptor 1; SSTR1; SS1R; SRIF-2
Click to Show/Hide
|
||||
| Target Type | Successful Target | ||||
| Gene Name | SSTR1 | ||||
| Biochemical Class | GPCR rhodopsin | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 2 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
1-(4-Aminobutyl)-9-benzyl-13-[(2R)-2-hydroxypropyl]-5-[2-(1H-indol-3-yl)ethyl]-1,5,9,13-tetrazacyclohexadecane-2,6,10,14-tetrone
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3218121
Click to Show/Hide
|
||||
| Activity |
Ki = 102000 nM
|
[1] | |||
| Compound Name |
1-(4-Aminobutyl)-8-benzyl-12-[(2R)-2-hydroxypropyl]-4-[2-(1H-indol-3-yl)ethyl]-1,4,8,12-tetrazacyclopentadecane-2,5,9,13-tetrone
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3218120
Click to Show/Hide
|
||||
| Activity |
Ki = 153000 nM
|
[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Synthesis and binding affinities for sst receptors of cyclic peptoid SRIF-mimetics. Medchemcomm. 2012;3:1531-5. | ||||
If You Find Any Error in Data or Bug in Web Service, Please Kindly Report It to Dr. Zhou and Dr. Zhang.