Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T89458 | Target Info | |||
| Target Name | HepG2 glucose transporter (SLC2A1) | ||||
| Synonyms |
Solute carrier family 2, facilitated glucose transporter member 1; HepG2 glucosetransporter; Glucose transporter type 1, erythrocyte/brain; GLUT1; GLUT-1
Click to Show/Hide
|
||||
| Target Type | Preclinical Target | ||||
| Gene Name | SLC2A1 | ||||
| Biochemical Class | Major facilitator | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 87 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Imidazo [1,2-a]pyridine compound 1
Click to Show/Hide
|
Patented | Compound Info | ||
| Synonyms |
PMID26882240-Compound-18
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
[(2R,3S,4S,5R)-3,4,5,6-Tetrahydroxyoxan-2-yl]methyl 4-[4-[bis(2-chloroethyl)amino]phenyl]butanoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4095994
Click to Show/Hide
|
||||
| Activity |
IC50 = 65000 nM
|
[2] | |||
| Compound Name |
(3R,4S,5R,6R)-6-(Hydroxymethyl)-4-(undec-10-enyloxy)-tetrahydro-2H-pyran-2,3,5-triol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL204300; BDBM50179102
Click to Show/Hide
|
||||
| Activity |
Ki = 98000 nM
|
[3] | |||
| Compound Name |
Chembl4290215
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL16261617; BDBM50527790
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4286532
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718968
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4281475
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718849
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4288783
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719043
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4283953
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719144
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4164091
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL20339793; BDBM50277387; AKOS008988719; 3-[(pyridin-4-ylmethylamino)methyl]phenol
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
Chembl4291571
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718883
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4293965
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719109
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
4-({6-Methyl-2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)piperazin-2-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4286284; SCHEMBL17718816; ZINC57273946; AKOS001304940; MCULE-4000083866; Z89087398
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4277005
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719088
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4290174
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718922
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
(2-Chlorophenyl)(4-{[2-(3-methoxyphenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl}piperazino)methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4290775; SCHEMBL17718825; ZINC98009878; AKOS021651412
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4281061
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718972
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4280066
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718854
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4279818
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718869
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4282894
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718864
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
3,3-Dimethyl-1-(4-{[2-(3-nitrophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl}piperazino)-1-butanone
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4292589; ZINC37384743; AKOS021737228
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4291853
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718873
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4285241
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718853
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4160688
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL20339305; BDBM50277369
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
Chembl4283657
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718988
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4290332
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719001
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4281884
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718945
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4282705
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719110
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
2,6-Dimethyl-4-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)morpholine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4285026; SCHEMBL17718818; AKOS032998730; MCULE-3124867547; Z103697440
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4285108
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719042
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4288878
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718904
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4171968
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL21500123; BDBM50277370; MCULE-6580806030
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
Chembl4285087
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
4-((6-bromo-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl)methyl)morpholine; 4-[[6-bromo-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]morpholine; SCHEMBL16246699
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4283210
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718933
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4293721
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718926
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4282115
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718973
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4285309
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718944
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4286446
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718876
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4283457
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718960
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4284054
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718893
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
6-Methyl-2-phenyl-3-(1,4-thiazinan-4-ylmethyl)imidazo[1,2-a]pyridine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
4-({6-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)thiomorpholine; MLS000721471; CHEMBL1324254; SCHEMBL17718803; HMS2615C16; KS-000036AK; MFCD04125116; ZINC20366664; AKOS005088844; 3N-545S; MCULE-9473852522; SMR000337111; SR-01000307780; SR-01000307780-1
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4292584
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718855
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4289978
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718921
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4280138
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718938
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4288094
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718895
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4282344
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719102
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4277550
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719060
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
2-(4-Chlorophenyl)-6-phenyl-3-(piperazin-1-ylmethyl)imidazo[1,2-a]pyridine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4280738; SCHEMBL12819033
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4285753
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718865
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4289439
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718871
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4288468
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719104
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4294333
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718898
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4278406
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718870
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4294938
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718986
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4283614
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719167
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
4-{[6-Chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl}thiomorpholine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
6-chloro-2-(4-chlorophenyl)-3-(1,4-thiazinan-4-ylmethyl)imidazo[1,2-a]pyridine; CHEMBL4289966; SCHEMBL16261616; ZINC20366650; AKOS005088741; 3N-513S; MCULE-6921563459; KS-0000369Z
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4289936
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719063
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4279963
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718850
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4165190
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL20338615; BDBM50277373
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
3-Methyl-1-(4-{[2-(3-nitrophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl}piperazino)-1-butanone
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4277214; SCHEMBL12819016; ZINC37385055; AKOS021743867
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4283125
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718861
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4289466
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719036
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
[4-(Tert-butyl)phenyl](4-{[2-(4-chlorophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl}piperazino)methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4286302; SCHEMBL17718828; ZINC98009880; AKOS021601181
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4281182
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718808
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
6-Chloro-2-(4-chlorophenyl)-3-(piperidinomethyl)imidazo[1,2-a]pyridine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
1-{[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine; MLS001195413; CHEMBL1480543; SCHEMBL16261619; HMS2851N20; ZINC4003070; AKOS005088901; 3N-515S; MCULE-9515962430; KS-000036A1; SMR000550582
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4292959
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17722629
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
(2-Chlorophenyl)(4-{[2-(4-chlorophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl}piperazino)methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4286507; SCHEMBL17718841; AKOS021973520; ZINC101664488
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4286844
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718874
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
4-{[2-(4-Chlorophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl]methyl}-N~1~-(4-methoxyphenyl)tetrahydro-1(2H)-pyrazinecarboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4291997; SCHEMBL17718842; AKOS021659568; ZINC103404695
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4290530
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718879
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4280977
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718884
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4286579
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718852
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4288373
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719050
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4278673
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718940
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4277963
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719051
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4278907
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718848
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4293579
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719041
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4286145
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718970
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4282384
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719147
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4279552
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718914
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4294162
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL16246753; tert-butyl 4-((2-(4-chlorophenyl)-6-phenylimidazo[1,2-a]pyridin-3-yl)methyl)piperazine-1-carboxylate
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4294955
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718862
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4280984
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718888
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Chembl4294011
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718889
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4283820
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17718959
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4278839
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719067
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
3-{[4-(2-Fluorophenyl)piperazino]methyl}-6-methyl-2-phenylimidazo[1,2-a]pyridine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
MLS000721492; CHEMBL1507648; SCHEMBL17718805; HMS2615P10; KS-000036AL; ZINC20366666; AKOS005088845; 3N-546S; MCULE-6835224964; SMR000337112
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Chembl4278601
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL17719103
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| Non Binders of This Target (in total, 3 non binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
(3R,4S,5S,6R)-6-((Undec-10-enyloxy)methyl)-tetrahydro-2H-pyran-2,3,4,5-tetraol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL249476; BDBM50216469
Click to Show/Hide
|
||||
| Activity |
Ki = 400000 nM
|
[3] | |||
| Compound Name |
(2R,3S,4S,5R,6R)-2-(Hydroxymethyl)-6-(undec-10-enyloxy)-tetrahydro-2H-pyran-3,4,5-triol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL248915; BDBM50216465
Click to Show/Hide
|
||||
| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
[(2R,3S,4R,5R)-4,5,6-Trihydroxy-2-(hydroxymethyl)oxan-3-yl] methanesulfonate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4066980
Click to Show/Hide
|
||||
| Activity |
IC50 = 32000000 nM
|
[2] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | US patent application no. 20160120863A1, SLC2A TRANSPORTER INHIBITORS | ||||
| REF 2 | Anticancer agents interacting with membrane glucose transporters. Medchemcomm. 2016 Sep 1;7(9):1716-1729. | ||||
| REF 3 | Interaction of O-(undec-10-en)-yl-D-glucose derivatives with the Plasmodium falciparum hexose transporter (PfHT). Bioorg Med Chem Lett. 2007 Sep 1;17(17):4934-7. | ||||
| REF 4 | Development of GLUT4-selective antagonists for multiple myeloma therapy. Eur J Med Chem. 2017 Oct 20;139:573-586. | ||||
If You Find Any Error in Data or Bug in Web Service, Please Kindly Report It to Dr. Zhou and Dr. Zhang.